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A one-pot conversion of artemisinin to arteether

Guo-Feng Wei, Zu-Liang Huang, Guang-Yu Pan, Xian-Jiu Liao, Li Qian


A one-pot preparation of anti-malaria arteether was developed. The influences of the trifluoroactic acid amount, reaction temperature, pH value as well as reaction time were studied in this paper.


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